Rh(III)-catalyzed cyclization reaction of azoles with alkynes: efficient synthesis of azole-fused-pyridines.

نویسندگان

  • Xuebing Chen
  • Youzhi Wu
  • Jinyi Xu
  • Hequan Yao
  • Aijun Lin
  • Yue Huang
چکیده

A Rh(iii)-catalyzed cyclization of azoles with alkynes has been developed. A variety of azole-fused-pyridines were obtained in good to excellent yields and regioselectivity. Both the C5 and the C4 position of azoles were suitable for the reaction.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 13 35  شماره 

صفحات  -

تاریخ انتشار 2015